KAPPE C O. 100 Years of the Biginelli Dihydropyrimidine Synthesis[J]. Tetrahedron, 1993, 49(32):6937-6963. doi: 10.1016/S0040-4020(01)87971-0
|
钟国清.无机及分析化学实验改革与绿色化实验教材建设[J].西南师范大学学报(自然科学版), 2018, 43(5):162-166.
|
章思规.精细有机化学品技术手册:下册[M].北京:科学出版社, 1992.
|
崔朋雷, 李晓慧, 张冬暖, 等.微波辐射下一锅法合成5-氰基-6-芳基硫脲嘧啶[J].西南大学学报(自然科学版), 2014, 36(7):79-83.
|
BIGINELLI P. Aldehyde-Urea Derivatives of Aceto-and Oxaloacetic Acids[J]. Gazzetta Chimica Italiana, 1893, 23(1):360-413.
|
SINGH K, ARORA D, POREMSKY E, et al. N1-Alkylated 3, 4-dihydropyrimidine-2(1H)-ones:Convenient One-Pot Selective Synthesis and Evaluation of Their Calcium Channel Blocking Activity[J]. European Journal of Medicinal Chemistry, 2009, 44(5):1997-2001. doi: 10.1016/j.ejmech.2008.10.002
|
ZALAVADIYA P, TALA S, AKBARI J, et al. Multi-Component Synthesis of Dihydropyrimidines by Iodine Catalyst at Ambient Temperature and in-vitro Antimycobacterial Activity[J]. Archiv Der Pharmazie, 2009, 342(8):469-475. doi: 10.1002/ardp.200800224
|
KAPPE C O. Microwave-Assisted High-Speed Parallel Synthesis of4-Aryl-3, 4-dihydropyrimidin-2(1H)-ones Using a Solventless Biginelli Condensation Protocol[J]. Synthesis, 1999, 1999(10):1799-1803. doi: 10.1055/s-1999-3592
|
SALEHI H, GUO Q X. Efficient Magnesium Bromide-Catalyzed One-Pot Synthesis of Substituted 1, 2, 3, 4-Tetrahydropyrimidin-2-ones Under Solvent-Free Conditions[J]. Chinese Journal of Chemistry, 2005, 23(1):91-97.
|
ISMAILI L, NADARADJANE A, NICOD L, et al. Synthesis and Antioxidant Activity Evaluation of New Hexahydropyrimido[5, 4-C] quinoline-2, 5-Diones and 2-Thioxohexahydropyrimido[5, 4-C] quinoline-5-Ones Obtained by Biginelli Reaction in Two Steps[J]. European Journal of Medicinal Chemistry, 2008, 43(6):1270-1275. doi: 10.1016/j.ejmech.2007.07.012
|
BESOLUK S, KUCUKISLAMOGLU M, NEBIOGLU M, et al. Solvent-Free Synthesis of Dihydropyrimidinones Catalyzed by Alumina Sulfuric Acid at Room Temperature[J]. Journal of the Iranian Chemical Society, 2008, 5(1):62-66. doi: 10.1007/BF03245816
|
ARIDOSS G, JEONG Y T. A Convenient One-Pot Biginelli Reaction Catalyzed by Y(OAc)3:An Improved Protocol for the Synthesis of 3, 4-Dihydropyrimidin-2(1H)-ones and Their Sulfur Analogues[J]. Bulletin of the Korean Chemical Society, 2010, 31(4):863-868. doi: 10.5012/bkcs.2010.31.04.863
|
LI W J, LIU S, HE P, et al. New Efficient Synthesis of Pyrimido[1, 6-c] Quinazolin-4-Ones by a Biginelli 3CC/Staudinger/Aza-Wittig Sequence[J]. Tetrahedron, 2010, 66(41):8151-8159. doi: 10.1016/j.tet.2010.08.046
|
CHENG Q F, WANG Q F, XU X Y, et al. Solvent-Free Synthesis of Monastrol Derivatives Catalyzed by NaHSO4[J]. Journal of Heterocyclic Chemistry, 2010:47(3):624-628.
|
MEMARIAN H R, RANJBAR M. Synthesis of Biginelli Compounds Using Cobalt Hydrogen Sulfate[J]. Journal of the Chinese Chemical Society, 2011, 58(4):522-527. doi: 10.1002/jccs.201190016
|
PUTATUNDA S, CHAKRABORTY S, GHOSH S, et al. Regioselective N1-Alkylation of 3, 4-dihydropyrimidine-2(1H)-ones:Screening of Their Biological Activities Against Ca2+-ATPase[J]. European Journal of Medicinal Chemistry, 2012, 54(8):223-231.
|
王敏, 姜宏旭, 张顺, 等.硝酸铋催化三组分"一锅法"合成N1-取代的3, 4-二氢嘧啶酮衍生物[J].化学研究与应用, 2017, 29(10):1584-1589. doi: 10.3969/j.issn.1004-1656.2017.10.023
|
王敏, 张顺, 姜宏旭.无溶剂条件下三氯化铁高效催化合成N1-取代的3, 4-二氢嘧啶-2(1H)-酮[J].渤海大学学报(自然科学版), 2017, 38(4):289-294. doi: 10.3969/j.issn.1673-0569.2017.04.002
|
KAPPE C O. A Reexamination of the Mechanism of the Biginelli Dihydropyrimidine Synthesis. Support for an N-Acyliminium Ion Intermediate1[J]. The Journal of Organic Chemistry, 1997, 62(21):7201-7204. doi: 10.1021/jo971010u
|